Bitolterol: Chemical Structure, Mechanism of Action, Uses & Side Effects

Chemical Structure/Formula:

• C28H31NO4

Structure of Bitolterol

Mechanism of Action:

• Bitolterol is a prodrug that is converted in the body to colterol, its active metabolite, which is a selective beta-2 adrenergic receptor agonist.

• It primarily causes bronchodilation by relaxing smooth muscle in the airways.

Uses:

• Its main use is in the treatment of asthma, where it helps to relieve symptoms like wheezing and shortness of breath.

Side Effects:

• Common side effects can include cough, nervousness, headache, tremor, and dryness of the mouth and throat.