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Butacaine

BP-S-5-MEDICINAL CHEMISTRY
1 min read

Structure

  • Butacaine is an amino benzoic acid derivative with a butyl ester group, providing effective local anesthetic properties.

  • Chemical Formula: C₁₀H₂₁N₃O₂

    formula of Butacaine
Structure of Butacaine
Structure of Butacaine

Mode of Action

  • Sodium Channel Blockade: Inhibits voltage-gated sodium channels, preventing nerve impulse propagation.

  • Membrane Stabilization: Reduces nerve excitability by altering membrane potential.

Uses

  • Local Anesthesia: Utilized in dental procedures, minor surgeries, and dermatological applications.

  • Topical Preparations: Applied to skin and mucous membranes for numbing before minor interventions.

  • Infiltration Anesthesia: Injected to numb specific areas during medical procedures.

Side Effects

  • Local Irritation: May cause redness, swelling, or itching at the application site.

  • Systemic Toxicity: Rare but possible with excessive use, leading to CNS and cardiovascular effects.


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