Structure (Cyproheptadine hydrochloride)
Cyproheptadine hydrochloride features a tricyclic structure with a dibenzocycloheptene core connected to a piperidine ring.
The hydrochloride salt enhances solubility.
Chemical Formula: C₂₂H₂₃ClN₂·HCl
Mode of Action
Functions as an H₁-antagonist with antiserotonergic and anticholinergic properties.
It blocks histamine and serotonin receptors.
Uses
Allergic Reactions: Effective in treating symptoms like sneezing, itching, and runny nose.
Appetite Stimulation: Used to increase appetite in conditions causing weight loss.
Migraine Prophylaxis: Utilized in preventing migraines due to its serotonergic antagonism.