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Diperodon

BP-S-5-MEDICINAL CHEMISTRY
1 min read

Structure

  • Diperodon is a synthetic amino benzoic acid derivative with a cyclohexylmethyl substituent, enhancing its local anesthetic potency.

  • Chemical Formula: C₁₀H₂₀N₂O₂

    formula of Diperodon
Structure of Diperodon
Structure of Diperodon

Mode of Action

  • Voltage-Gated Sodium Channel Inhibition: Blocks sodium influx, preventing nerve impulse transmission.

  • Membrane Stabilization: Reduces nerve excitability by stabilizing neuronal membranes.

Uses

  • Local Anesthesia: Used in dental procedures, minor surgical interventions, and dermatological applications.

  • Topical Preparations: Applied to skin and mucous membranes for temporary numbing.

  • Ophthalmic Anesthesia: Employed in eye surgeries for effective corneal numbing.

Side Effects

  • Local Reactions: Redness, swelling, or irritation at the application site.

  • Systemic Toxicity: Potential CNS and cardiovascular effects with excessive use.


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