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Meprylcaine

Structure

  • Meprylcaine is a synthetic local anesthetic with a diethylaminoethyl substituent attached to a benzamide core.

  • Chemical Formula: C₁₁H₂₂N₂O

    Formula of Meprylcaine
Structure of Meprylcaine
Structure of Meprylcaine

Mode of Action

  • Sodium Channel Blockade: Inhibits nerve impulse transmission by blocking voltage-gated sodium channels.

  • Extended Duration: Provides longer-lasting anesthesia compared to simpler local anesthetics.

Uses

  • Local Anesthesia: Used in minor surgical procedures and dental applications.

  • Topical Preparations: Applied to mucous membranes for numbing before procedures.

Side Effects

  • Central Nervous System Effects: Dizziness, tremors, and seizures with excessive use.

  • Cardiovascular Toxicity: Hypotension and arrhythmias in high doses.


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